SCHEMBL8766829

SCHEMBL8766829

CCCOc1cnc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)nc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 1/20 0.37
CHRM1 P11229 1/20 0.36
HTR2A P28223 1/20 0.36
MCHR1 Q99705 1/20 0.36
GRM5 P41594 3/20 0.35
MAPT P10636 2/20 0.34
ACACB O00763 6/20 0.33
ALDH1A1 P00352 1/20 0.33
KDM1A O60341 1/20 0.32
PTPN7 P35236 1/20 0.32
DUSP3 P51452 1/20 0.32
CHRNA7 P36544 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9433084 0.91 CHRNA7 (0.39) NPC1RAB9ASMN1; SMN2HSD17B10CHRM1
SCHEMBL8766245 0.86 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2HSD17B10KDM4E
SCHEMBL8766249 0.85 RARA (0.41) CHRM1HTR2AMCHR1GRM5ACACB
SCHEMBL8766815 0.84 KDM1A (0.32) KDM4EGRM5MAPTALDH1A1KDM1A
SCHEMBL8767583 0.84 NPC1 (0.39) NPC1RAB9ASMN1; SMN2HSD17B10GRM5
SCHEMBL8767204 0.84 RXRA (0.36) GRM5
SCHEMBL8766253 0.82 RARB (0.38) NPC1RAB9ASMN1; SMN2HSD17B10KDM4E
SCHEMBL8767188 0.81 RARB (0.45) NPC1RAB9ASMN1; SMN2HSD17B10KDM4E
SCHEMBL8766819 0.81 RARB (0.43) NPC1RAB9ASMN1; SMN2HSD17B10KDM4E
SCHEMBL9469740 0.80 ACACB (0.46) GRM5ACACBCHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed