SCHEMBL876752

SCHEMBL876752

Nc1cc(N2C=CON2)ccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.36
NOS2 P35228 4/20 0.36
NOS1 P29475 3/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CDC7 O00311 1/20 0.34
CDK2 P24941 1/20 0.34
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB1 P18505 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
GABRB2 P47870 2/20 0.33
GABRA4 P48169 2/20 0.33
GABRE P78334 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8931619 0.71 LGMN (0.37) KDM4EMEN1KMT2A
SCHEMBL6780438 0.67 ADRB1 (0.49) NOS3NOS2KDM4ECDC7CDK2
SCHEMBL14858374 0.66 NOS3 (0.46) NOS3NOS2NOS1KDM4EMEN1
SCHEMBL7382496 0.66 NPC1 (0.43) KDM4EMEN1KMT2A
Ammonia Solution, Strong SCHEMBL1065028 0.65 CFTR (0.33)
SCHEMBL28047779 0.63 MAPT (0.50) NOS3NOS2NOS1KDM4EMEN1
SCHEMBL114416 0.62 LGMN (0.53) CDK2
SCHEMBL6643085 0.62 ADRB2 (0.56)
SCHEMBL30321663 0.62 LGMN (0.53) CDK2
SCHEMBL16212228 0.62 HRH4 (0.47) NOS3NOS2NOS1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619190-A1 SUBSTITUTED OXADIAZOLE COMPOUNDS AND THEIR USE AS S1P1 AGONISTS Bristol-Myers Squibb Company (US) 2013-07-31 EP claimed
WO-2012040532-A1 SUBSTITUTED OXADIAZOLE COMPOUNDS AND THEIR USE AS S1P1 AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-29 WO claimed