SCHEMBL8772012

SCHEMBL8772012

NC(=O)Cc1c(F)ccc([N+](=O)[O-])c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.40
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HIF1A Q16665 1/20 0.35
TTR P02766 1/20 0.34
LMNA P02545 3/20 0.34
RECQL P46063 1/20 0.34
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CES2 O00748 1/20 0.33
ABCB11 O95342 1/20 0.33
GLA P06280 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CHRM1 P11229 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
TBXA2R P21731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772070 0.88 AR (0.42) ARATMTDP1ALDH1A1HIF1A
SCHEMBL2975400 0.82 ATM (0.40) ATMTDP1ALDH1A1HIF1ALMNA
SCHEMBL8772047 0.77 ICMT (0.32) ALDH1A1
SCHEMBL27816496 0.77 LMNA (0.40) ATMTDP1ALDH1A1HIF1ALMNA
SCHEMBL30625901 0.76 ALDH1A1 (0.43) TDP1ALDH1A1LMNACYP3A4CYP1A2
SCHEMBL8771996 0.73 AR (0.44) ARATMTDP1ALDH1A1HIF1A
SCHEMBL27891591 0.70 ALDH1A1 (0.43) ARATMTDP1ALDH1A1HIF1A
SCHEMBL30153092 0.70 ALDH1A1 (0.45) ARATMTDP1ALDH1A1HIF1A
SCHEMBL15971307 0.70 TDP1 (0.45) ARATMTDP1ALDH1A1HIF1A
SCHEMBL3131783 0.70 LMNA (0.54) ALDH1A1HIF1ALMNARECQLHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686492-A NMR DIAGNOSTIC AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 1997-11-11 US disclosed
EP-0799197-A1 DISUBSTITUTED P-FLUOROBENZOLSULFONAMIDES AND THEIR USE IN NMR DIAGNOSTICS SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-08 EP disclosed
WO-1996019447-A1 DISUBSTITUTED P-FLUOROBENZOLSULFONAMIDES AND THEIR USE IN NMR DIAGNOSTICS SCHERING AKTIENGESELLSCHAFT (DE) 1996-06-27 WO disclosed