SCHEMBL8772047

SCHEMBL8772047

NC(=O)Cc1c(F)ccc(N)c1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ICMT O60725 1/20 0.32
CA2 P00918 1/20 0.32
HDAC1 Q13547 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
SIRT1 Q96EB6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8915526 0.81 GAA (0.40) KDM4EALDH1A1HSD17B10
SCHEMBL7245085 0.80 CA2 (0.36) ICMTCA2HDAC1HDAC6ALDH1A1
SCHEMBL8772012 0.77 AR (0.40) ALDH1A1
SCHEMBL12984831 0.72 CES2 (0.40) ICMTCA2
SCHEMBL8772056 0.71 P2RX7 (0.45)
SCHEMBL6390159 0.70 MAPK8 (0.49) CA2KDM4E
SCHEMBL8913345 0.70 ADRA1B (0.35) CA2ALDH1A1
Hydrochloric Acid SCHEMBL28042671 0.68 ALDH1A1 (0.35) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9747729 0.68 ALDH1A1 (0.36) ALDH1A1
SCHEMBL7871395 0.68 ALDH1A1 (0.36) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686492-A NMR DIAGNOSTIC AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 1997-11-11 US disclosed
EP-0799197-A1 DISUBSTITUTED P-FLUOROBENZOLSULFONAMIDES AND THEIR USE IN NMR DIAGNOSTICS SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-08 EP disclosed
WO-1996019447-A1 DISUBSTITUTED P-FLUOROBENZOLSULFONAMIDES AND THEIR USE IN NMR DIAGNOSTICS SCHERING AKTIENGESELLSCHAFT (DE) 1996-06-27 WO disclosed