SCHEMBL8772253

SCHEMBL8772253

OCc1cccc([C@@H](O)Cc2cccc(Br)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
LTB4R Q15722 5/20 0.35
PRKCI P41743 1/20 0.33
ENPP2 Q13822 1/20 0.33
CDK8 P49336 1/20 0.32
ROCK2 O75116 1/20 0.32
ADRB2 P07550 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
CYSLTR1 Q9Y271 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772241 1.00 NOS1 (0.44) NOS1NOS2LTB4RPRKCIENPP2
SCHEMBL8772160 0.74 LTB4R (0.47) LTB4RCDK8ADRB2CYSLTR1
SCHEMBL8772152 0.74 LTB4R (0.47) LTB4RCDK8ADRB2CYSLTR1
SCHEMBL7144095 0.73 PNMT (0.54) NOS1NOS2PRKCIENPP2ROCK2
SCHEMBL8772170 0.72 LTB4R (0.48) LTB4R
SCHEMBL8772180 0.72 LTB4R (0.48) LTB4R
SCHEMBL105003 0.70
SCHEMBL29811249 0.70
SCHEMBL24015105 0.70 LMNA (0.55) NOS1NOS2PRKCIENPP2ADRB2
SCHEMBL1249740 0.70 NOS2 (0.41) NOS2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0801061-A2 Leucotrien-B4 derivatives, process for their preparation and their use as medicaments SCHERING AKTIENGESELLSCHAFT (DE) 1997-10-15 EP disclosed
US-5614634-A Leukotriene-B4 derivatives, process for their production and their use as pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1997-03-25 US disclosed
US-5440044-A Leukotriene-B4 derivatives, process for their production and their use as pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1995-08-08 US disclosed
EP-0477311-A1 NEW LEUCOTRIENE B 4? DERIVATIVES, METHODS OF PREPARING THEM AND THEIR USE AS DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1992-04-01 EP disclosed
WO-1991014676-A1 NEW LEUCOTRIENE B4 DERIVATIVES, METHODS OF PREPARING THEM AND THEIR USE AS DRUGS SCHERING AKTIENGESELLSCHAFT BERLIN UND BERGKAMEN (DE) 1991-10-03 WO disclosed