SCHEMBL8772491

SCHEMBL8772491

O=C1CC(S(=O)(=O)c2ccccc2)N1CCCCCCc1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.42
KCNH2 Q12809 2/20 0.42
PSEN1 P49768 3/20 0.40
PSEN2 P49810 3/20 0.40
APH1B Q8WW43 3/20 0.40
NCSTN Q92542 3/20 0.40
APH1A Q96BI3 3/20 0.40
PSENEN Q9NZ42 3/20 0.40
ALDH1A1 P00352 2/20 0.40
FKBP1A P62942 1/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR2C P28335 1/20 0.38
POLB P06746 1/20 0.38
CCR3 P51677 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772454 0.85 POLB (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8438916 0.83 PLAAT3 (0.45) ALDH1A1TP53MEN1KMT2APOLB
SCHEMBL8772476 0.81 ALDH1A1 (0.46) KCNH2ALDH1A1POLBSIGMAR1TDP1
SCHEMBL8439355 0.77 GSK3A (0.44) ALDH1A1TP53GAAMEN1KMT2A
SCHEMBL8104154 0.76 FAAH (0.44) HTR2AKCNH2TP53MEN1KMT2A
SCHEMBL8772537 0.74 POLB (0.40) ALDH1A1POLBCCR3SIGMAR1GSK3A
SCHEMBL8772474 0.74 POLB (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8772449 0.74 CYP1A2 (0.42) HTR2AALDH1A1FKBP1ATP53GAA
SCHEMBL8439468 0.72 HTR2A (0.40) HTR2AKCNH2ALDH1A1MEN1KMT2A
SCHEMBL8441542 0.71 ALDH1A1 (0.52) KCNH2ALDH1A1MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799200-A1 SUBSTITUTED AZETIDIN-2-ONES FOR TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-10-08 EP disclosed