SCHEMBL8772898

SCHEMBL8772898

CSC(N)=NCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.60
GRIN2B Q13224 12/20 0.55
GRIN1 Q05586 8/20 0.55
GRIN2D O15399 3/20 0.55
GRIN3B O60391 3/20 0.55
GRIN2A Q12879 3/20 0.55
GRIN2C Q14957 3/20 0.55
GRIN3A Q8TCU5 3/20 0.55
SIGMAR1 Q99720 2/20 0.55
HRH4 Q9H3N8 2/20 0.43
HRH3 Q9Y5N1 2/20 0.43
GAA P10253 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SCN2A Q99250 1/20 0.43
IDO1 P14902 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL10591785 0.98 NOS2 (0.58) NOS2GRIN2BGRIN1GRIN2DGRIN3B
SCHEMBL15041111 0.81 NOS2 (0.58) NOS2GRIN2BGRIN1GRIN2DGRIN3B
SCHEMBL4646866 0.81 NOS2 (0.58) NOS2GRIN2BGRIN1GRIN2DGRIN3B
SCHEMBL9062832 0.80 NOS1 (0.68) NOS2GRIN2BGRIN1GRIN2DGRIN3B
Iodide SCHEMBL11389805 0.79 NOS3 (0.56) NOS2GRIN2BGRIN1HRH4HRH3
Bromide SCHEMBL11806754 0.79 NOS2 (0.59) NOS2GRIN2BGRIN1GRIN2DGRIN3B
SCHEMBL14291059 0.77 NOS2 (0.96) NOS2GRIN2BGRIN1GRIN2DGRIN3B
SCHEMBL20675953 0.77 NOS2 (0.96) NOS2GRIN2BGRIN1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL10516683 0.77 HTR3A (0.66) NOS2GRIN2BGRIN1HRH4HRH3
SCHEMBL45769 0.76 GRIN2B (0.68) NOS2GRIN2BGRIN1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625967-B1 N,N'-SUBSTITUTED IMIDOCARBONIMIDIC DIAMIDES DERIVED FROM HYDROXYLAMINES JACOBUS PHARMA CO INC (US) 1997-08-27 EP disclosed
WO-1995028377-A1 GUANIDINE COMPOUNDS AS REGULATORS OF NITRIC OXIDE SYNTHASE ABBOTT LABORATORIES (US) 1995-10-26 WO disclosed
EP-0625967-A1 N,N'-SUBSTITUTED IMIDOCARBONIMIDIC DIAMIDES DERIVED FROM HYDROXYLAMINES. JACOBUS PHARMA CO INC (US) 1994-11-30 EP disclosed
US-5322858-A Antimicrobial, antiparasitic agents JACOBUS PHARMACEUTICAL CO. INC. (US) 1994-06-21 US disclosed
WO-1993016037-A1 N,N'-SUBSTITUTED IMIDOCARBONIMIDIC DIAMIDES DERIVED FROM HYDROXYLAMINES JACOBUS PHARMACEUTICAL CO., INC. (US) 1993-08-19 WO disclosed