SCHEMBL8774813

SCHEMBL8774813

CCCCCOc1ccc(CCc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP1 P29466 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SLCO1B3 Q9NPD5 1/20 0.42
SLCO1B1 Q9Y6L6 1/20 0.42
NR5A1 Q13285 1/20 0.41
PKM P14618 1/20 0.40
LTA4H P09960 1/20 0.40
S1PR4 O95977 3/20 0.40
S1PR1 P21453 3/20 0.40
S1PR3 Q99500 3/20 0.40
S1PR5 Q9H228 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8775001 0.97 PKM (0.42) MEN1KMT2AUSP2ALDH1A1LMNA
SCHEMBL8774330 0.96 CYP3A4 (0.43) MEN1KMT2AUSP2ALDH1A1LMNA
SCHEMBL8774925 0.94 CYP2D6 (0.46) MEN1KMT2AUSP2ALDH1A1LMNA
SCHEMBL8774833 0.92 LMNA (0.44) ALDH1A1LMNASMN1; SMN2
SCHEMBL8774847 0.88 ACACB (0.43) MEN1KMT2AALDH1A1LMNACYP3A4
SCHEMBL8774796 0.86 NQO1 (0.41) ALDH1A1LMNASMN1; SMN2
SCHEMBL8774823 0.86 HTR2A (0.46) ALDH1A1LMNACYP3A4
SCHEMBL8774041 0.85 HTR2A (0.49) ALDH1A1LMNACYP3A4
SCHEMBL8774498 0.84 HTR2A (0.40) ALDH1A1LMNACYP3A4SMN1; SMN2
SCHEMBL9161261 0.83 MEN1 (0.43) MEN1KMT2AUSP2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed