SCHEMBL8774719

SCHEMBL8774719

CCCCCCCc1ccc(C#Cc2cnc(F)c(F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.44
TSHR P16473 1/20 0.44
HTR2A P28223 1/20 0.44
FFAR1 O14842 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RARB P10826 3/20 0.41
RARA P10276 1/20 0.41
RARG P13631 1/20 0.41
ESR1 P03372 2/20 0.41
ADRA2A P08913 2/20 0.41
ADORA3 P0DMS8 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8775133 0.95 HSD17B10 (0.49) HSD17B10TSHRHTR2AFFAR1KDM4E
SCHEMBL8774677 0.94 FFAR1 (0.43) HSD17B10TSHRHTR2AFFAR1KDM4E
SCHEMBL8774460 0.91 HSD17B10 (0.43) HSD17B10TSHRFFAR1KDM4EALDH1A1
SCHEMBL8774897 0.89 FFAR1 (0.45) HSD17B10FFAR1RAB9ASMN1; SMN2TP53
SCHEMBL8774819 0.85 FFAR1 (0.43) HSD17B10TSHRFFAR1MAPTRAB9A
SCHEMBL8774154 0.83 EGLN1 (0.47) FFAR1
SCHEMBL8774700 0.82 KDM4E (0.47) HSD17B10TSHRKDM4EALDH1A1HPGD
SCHEMBL8774634 0.82 KDM4E (0.43) HSD17B10KDM4EALDH1A1HPGDRAB9A
SCHEMBL9158759 0.82 HSD17B10 (0.48) HSD17B10TSHRHTR2AFFAR1KDM4E
SCHEMBL8774239 0.81 HTR2A (0.50) HSD17B10HTR2AKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed