SCHEMBL8774239

SCHEMBL8774239

CCCCCCCc1ccc(CCc2cnc(F)c(F)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.50
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
USP2 O75604 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
ESR1 P03372 2/20 0.46
ADRA2A P08913 2/20 0.46
ADORA3 P0DMS8 2/20 0.46
TACR2 P21452 2/20 0.46
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
SLC6A3 Q01959 2/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774406 0.94 RARB (0.50) HTR2AKDM4EALDH1A1HSD17B10MAPT
SCHEMBL8774481 0.94 NFKB1 (0.44) HTR2AKDM4EALDH1A1HSD17B10MAPT
SCHEMBL8774784 0.89 RAB9A (0.46) KDM4EALDH1A1HSD17B10MAPTRAB9A
SCHEMBL8775147 0.87 NPC1 (0.47) HTR2AHSD17B10MAPTRAB9ASMN1; SMN2
SCHEMBL8774858 0.85 MEN1 (0.44) ALDH1A1MAPTRAB9ASMN1; SMN2MEN1
SCHEMBL8774557 0.85 RARB (0.57) HTR2AKDM4EALDH1A1HSD17B10MAPT
SCHEMBL8774898 0.85 RARB (0.57) HTR2AKDM4EALDH1A1HSD17B10MAPT
SCHEMBL8774178 0.85 CYP3A4 (0.43) ALDH1A1HSD17B10MAPTRAB9ASMN1; SMN2
SCHEMBL8774942 0.85 RARB (0.57) HTR2AKDM4EALDH1A1HSD17B10MAPT
SCHEMBL8774709 0.85 RARB (0.57) HTR2AKDM4EALDH1A1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed