SCHEMBL8774833

SCHEMBL8774833

CCCOc1ccc(CCc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HTT P42858 2/20 0.43
HSD17B10 Q99714 1/20 0.43
DHFR P00374 1/20 0.42
MAPT P10636 3/20 0.40
ALDH1A1 P00352 2/20 0.40
SLC5A1 P13866 1/20 0.40
SLC5A2 P31639 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PLA2G4A P47712 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA7 P36544 1/20 0.40
C3AR1 Q16581 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774847 0.96 ACACB (0.43) LMNAL3MBTL1HTTHSD17B10DHFR
SCHEMBL8775001 0.94 PKM (0.42) LMNAALDH1A1CHRNB4CHRNA3CHRNA7
SCHEMBL8774813 0.92 MEN1 (0.42) LMNAALDH1A1SMN1; SMN2
SCHEMBL8774925 0.91 CYP2D6 (0.46) LMNAL3MBTL1HSD17B10MAPTALDH1A1
SCHEMBL8774796 0.89 NQO1 (0.41) LMNADHFRALDH1A1SLC5A1SLC5A2
SCHEMBL8774330 0.89 CYP3A4 (0.43) LMNAL3MBTL1MAPTALDH1A1RAB9A
SCHEMBL8774157 0.85 RAB9A (0.39) LMNAL3MBTL1HSD17B10DHFRMAPT
SCHEMBL8774829 0.84 RAB9A (0.36) HSD17B10MAPTALDH1A1NPC1RAB9A
SCHEMBL8774180 0.82 TAAR1 (0.47) L3MBTL1HTTMAPTALDH1A1HPGD
SCHEMBL9158863 0.82 LMNA (0.46) LMNAL3MBTL1HTTHSD17B10DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed