SCHEMBL8779023

SCHEMBL8779023

CCCCOc1ccc(O)c(OC(=O)NC(=O)CN)n1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
PDE4A P27815 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
FAAH O00519 9/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
SMPD1 P17405 1/20 0.34
MMP1 P03956 1/20 0.34
PRSS1 P07477 1/20 0.34
ACR P10323 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779161 0.96 SMPD1 (0.39) CYP1A2CYP2D6SMN1; SMN2HDAC6FAAH
SCHEMBL8779132 0.94 ACACB (0.34) FAAHMAPTCA12CA1CA2
SCHEMBL8779296 0.89 MEN1 (0.33) KMT2A
SCHEMBL8779424 0.89 MAPK8 (0.37) KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL8779185 0.86 ACACB (0.37) KMT2A
SCHEMBL8779211 0.85 MEN1 (0.40) KDM4ECYP1A2SMN1; SMN2KMT2AMAPT
SCHEMBL8779357 0.84 GPR88 (0.32)
SCHEMBL8779178 0.83 PRKD3 (0.33) KDM4ESMN1; SMN2MAPTCA2SMPD1
SCHEMBL8786050 0.82 MEN1 (0.38) PDE4AFAAHKMT2AMAPTSMPD1
SCHEMBL8779309 0.81 L3MBTL1 (0.39) CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed