SCHEMBL8779246

SCHEMBL8779246

NCC(=O)NC(=O)Oc1nccc(OCc2ccc(C(F)(F)F)cc2)c1O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.43
PPIA P62937 1/20 0.39
PTPN1 P18031 4/20 0.39
PTPN2 P17706 2/20 0.39
PTPN6 P29350 2/20 0.39
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SPHK2 Q9NRA0 1/20 0.37
SPHK1 Q9NYA1 1/20 0.37
NR3C2 P08235 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
KDM5A P29375 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
FFAR1 O14842 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779187 0.92 MRGPRX4 (0.37) MAOBPPIAPTPN1PTPN2PTPN6
SCHEMBL8779285 0.89 KDM4E (0.40) MAOBALDH1A1
SCHEMBL8779269 0.89 L3MBTL1 (0.46) MAOBPPIAPTPN1ALDH1A1SPHK2
SCHEMBL8779331 0.89 MMP1 (0.41) MAOBRXRARXRBRXRGMRGPRX4
SCHEMBL8779168 0.87 SMN1; SMN2 (0.40) MAOBPPIAALDH1A1
SCHEMBL8779406 0.87 LTA4H (0.44) PPIA
SCHEMBL8785593 0.87 MAOB (0.41) MAOBPPIAPTPN1PTPN2PTPN6
SCHEMBL8785286 0.86 PPIA (0.49) MAOBPPIAPTPN1PTPN2PTPN6
SCHEMBL8779238 0.85 CYP1A2 (0.36) ALDH1A1
SCHEMBL8779316 0.85 MME (0.39) MAOBPPIAPTPN1PTPN2PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed