SCHEMBL8779331

SCHEMBL8779331

NCC(=O)NC(=O)Oc1nccc(OCc2ccc(OC(F)(F)F)cc2)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP14 P50281 1/20 0.41
ADAM17 P78536 1/20 0.41
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
MAPK8 P45983 1/20 0.38
MRGPRX4 Q96LA9 2/20 0.38
NLRP3 Q96P20 1/20 0.37
MAOB P27338 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
HTR2C P28335 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779246 0.89 MAOB (0.43) MRGPRX4MAOBRXRARXRBRXRG
SCHEMBL8787806 0.87 MMP1 (0.42) MMP1MMP2MMP9MMP14ADAM17
SCHEMBL8779285 0.86 KDM4E (0.40) MAOBMEN1KMT2ASMN1; SMN2
SCHEMBL8779265 0.85 TRPV1 (0.38) MMP1MMP2MMP9MMP14ADAM17
SCHEMBL8779168 0.84 SMN1; SMN2 (0.40) MAOBMEN1KMT2ASMN1; SMN2
SCHEMBL8779406 0.84 LTA4H (0.44) SMN1; SMN2TDP1
SCHEMBL8883592 0.84 TLR7 (0.43) MMP1MMP2MMP9MMP14ADAM17
SCHEMBL8779187 0.83 MRGPRX4 (0.37) MRGPRX4MAOB
SCHEMBL8779238 0.81 CYP1A2 (0.36) SMN1; SMN2
SCHEMBL8779269 0.80 L3MBTL1 (0.46) MRGPRX4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed