SCHEMBL8780460

SCHEMBL8780460

CCC(C)c1cc(Cc2ccc(C#N)cc2)c2ccccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
NTRK1 P04629 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
MAPK1 P28482 2/20 0.38
PKM P14618 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ABCG2 Q9UNQ0 3/20 0.37
ABCB1 P08183 1/20 0.37
ADAM17 P78536 1/20 0.36
CYP2A6 P11509 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
ALOX5AP P20292 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CTNNB1 P35222 1/20 0.36
TCF7L2 Q9NQB0 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6630276 0.77 ADAM17 (0.45) SMN1; SMN2MAPK1RXFP1ADAM17MEN1
SCHEMBL8780501 0.76 MEN1 (0.42) CYP11B1CYP11B2NTRK1SMN1; SMN2ABCG2
SCHEMBL25523507 0.74 CYP1A2 (0.53) SMN1; SMN2RXFP1POLBKMT2AALDH1A1
SCHEMBL8780490 0.73 KDR (0.36) NTRK1SMN1; SMN2ABCG2CYP2A6USP2
SCHEMBL6630282 0.70 ADAM17 (0.46) MAPK1ADAM17CYP2A6POLBMEN1
SCHEMBL7849358 0.70 TLR8 (0.42) POLBMEN1KMT2AALDH1A1ATM
SCHEMBL21027636 0.68 TNKS2 (0.44) SMN1; SMN2RXFP1ADAM17MEN1KMT2A
SCHEMBL7984282 0.67 MAPK1 (0.53) NTRK1MAPK1ABCG2USP2MEN1
SCHEMBL6487073 0.67 ADAM17 (0.45) SMN1; SMN2RXFP1ADAM17POLBMEN1
SCHEMBL7979804 0.66 L3MBTL1 (0.56) MAPK1RXFP1ABCG2ABCB1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP disclosed
EP-0498722-A1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1992-08-12 EP disclosed