SCHEMBL8782842

SCHEMBL8782842

NC(=O)N(O)CCNC(=O)c1cccc(S(=O)(=O)c2ccc(F)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.54
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 1/20 0.47
LOX P28300 2/20 0.46
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
NAMPT P43490 1/20 0.43
EPHX2 P34913 5/20 0.43
ALOX5 P09917 3/20 0.43
HSD17B10 Q99714 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GAA P10253 1/20 0.40
AKR1C3 P42330 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8783392 0.89 MEN1 (0.47) PKMMEN1KMT2AALDH1A1MAPK1
SCHEMBL8942652 0.84 PKM (0.44) PKMMEN1KMT2AALDH1A1MAPK1
SCHEMBL29280967 0.75 HTR2A (0.68) ALDH1A1HTR2AHTR2CGAAAKR1C3
SCHEMBL29280971 0.74 HDAC6 (0.49) PKMMEN1KMT2AALDH1A1NAMPT
SCHEMBL8783039 0.73 TDP1 (0.49) MEN1KMT2AALDH1A1EPHX2ALOX5
SCHEMBL8942817 0.73 GAA (0.42) PKMMEN1KMT2ALOXNAMPT
SCHEMBL8783271 0.72 SIGMAR1 (0.57) MEN1KMT2AALDH1A1HSD17B10NPC1
SCHEMBL999837 0.71 CXCR2 (0.57) ALDH1A1HTR2AHTR2CAKR1C3
SCHEMBL8783294 0.71 MEN1 (0.57) PKMMEN1KMT2AALDH1A1EPHX2
SCHEMBL8783388 0.70 ALOX5 (0.48) MEN1KMT2AALDH1A1EPHX2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0595995-B1 ARYLAMIDOALKYL- AND ARYLAMINOALKYL-N-HYDROXYUREA COMPOUNDS AND -N-HYDROXYFORMAMIDE DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LAB (US) 1997-01-15 EP disclosed
US-5514702-A Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1996-05-07 US disclosed