SCHEMBL8795290

SCHEMBL8795290

O=S(=O)(c1ccc(OCCCc2c[nH]cn2)cc1)c1ccc(OCCCc2c[nH]cn2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HRH3 Q9Y5N1 6/20 0.40
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
CA7 P43166 3/20 0.40
TSHR P16473 2/20 0.40
KCNH2 Q12809 4/20 0.39
GAA P10253 2/20 0.38
PKM P14618 2/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.37
RECQL P46063 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
CA4 P22748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4379847 0.93 HTR2A (0.42) ALDH1A1HRH3CA12CA1CA2
SCHEMBL4383470 0.85 LMNA (0.45) ALDH1A1CA12CA1CA2CA9
Oxalic Acid SCHEMBL7991431 0.80 SMN1; SMN2 (0.45) ALDH1A1LMNAL3MBTL1
SCHEMBL4380966 0.80 NQO1 (0.45) ALDH1A1HRH3TSHRKCNH2LMNA
SCHEMBL7961327 0.80 RAB9A (0.43) ALDH1A1HRH3KCNH2LMNA
SCHEMBL7987297 0.80 HRH3 (0.54) ALDH1A1HRH3KCNH2LMNAMAPK1
SCHEMBL4384169 0.79 ALDH1A1 (0.48) ALDH1A1CA9KCNH2LMNAL3MBTL1
SCHEMBL4376189 0.78 KCNH2 (0.37) ALDH1A1HRH3KCNH2LMNA
SCHEMBL4386689 0.78 LMNA (0.45) ALDH1A1HRH3TSHRKCNH2LMNA
SCHEMBL4376133 0.78 HRH3 (0.46) HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760811-A1 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H 3? (ANT)AGONISTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-03-12 EP claimed
EP-0594702-B1 SUBSTITUTED INDOLES AS ANTI-AIDS PHARMACEUTICALS UPJOHN CO (US) 1997-01-29 EP claimed
WO-1996029315-A2 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H3 (ANT)AGONISTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1996-09-26 WO claimed