SCHEMBL8799009

SCHEMBL8799009

COC(OC)C1(C)C=C(c2cccnc2)c2cc(NS(=O)(=O)c3ccccc3)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
BRD4 O60885 2/20 0.41
PIK3CA P42336 2/20 0.40
HPGD P15428 1/20 0.39
CYP17A1 P05093 3/20 0.38
GAA P10253 1/20 0.38
ALDH1A1 P00352 2/20 0.38
ALPL P05186 1/20 0.38
KDR P35968 1/20 0.38
GSK3B P49841 1/20 0.38
NAMPT P43490 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAP2K7 O14733 1/20 0.36
MAP2K4 P45985 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798430 0.90 IMPDH2 (0.43) BRD4HPGDCYP17A1ALDH1A1LMNA
SCHEMBL9233065 0.86 CYP11B1 (0.44) CYP11B1CYP11B2KEAP1NFE2L2BRD4
SCHEMBL8797664 0.85 HTR6 (0.37) NAMPTLMNA
SCHEMBL8798345 0.84 BRD4 (0.42) BRD4HPGDCYP17A1GAAALDH1A1
SCHEMBL9086171 0.79 KCNH2 (0.42) CYP11B1CYP11B2HPGDCYP17A1GAA
SCHEMBL8797782 0.76 CYP11B2 (0.40) CYP11B1CYP11B2CYP17A1
SCHEMBL9230527 0.75 IMPDH2 (0.48) BRD4HPGDALDH1A1LMNASMN1; SMN2
SCHEMBL8796818 0.75 KDM4E (0.33) PIK3CAHPGDGAAALDH1A1NAMPT
SCHEMBL8797621 0.75 BRD4 (0.40) BRD4HPGDCYP17A1ALDH1A1LMNA
SCHEMBL8796991 0.74 POLB (0.40) CYP11B1CYP11B2KDRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514942-B1 Novel benzopyran derivatives and processes for the preparation thereof KOREA RES INST CHEM TECH (KR) 1997-03-05 EP disclosed
US-5493029-A USEFUL IN TREATING ASTHMA AND HYPERTENSION KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1996-02-20 US disclosed
US-5300511-A Spiro-benzopyran derivatives and useful for treating asthma and hypertension KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1994-04-05 US disclosed
EP-0514942-A1 Novel benzopyran derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1992-11-25 EP disclosed