SCHEMBL8797664

SCHEMBL8797664

COC(OC)C1(C)C=C(c2cccnc2)c2cc(S(=O)(=O)c3ccccc3)ccc2O1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.37
NAMPT P43490 9/20 0.36
PTGS2 P35354 1/20 0.35
CYP2C9 P11712 2/20 0.33
BACE1 P56817 1/20 0.33
KCNH2 Q12809 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
PKM P14618 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796818 0.89 KDM4E (0.33) HTR6NAMPTPTGS2
SCHEMBL8799009 0.85 CYP11B1 (0.43) NAMPTLMNA
SCHEMBL9087771 0.85 HTR6 (0.42) HTR6NAMPTPTGS2CYP2C9BACE1
SCHEMBL8796821 0.83 HTR6 (0.33) HTR6NAMPTPTGS2
SCHEMBL9067938 0.82 CYP19A1 (0.41) PTGS2
SCHEMBL9086171 0.81 KCNH2 (0.42) PTGS2BACE1KCNH2CYP1A2CYP3A4
SCHEMBL8797782 0.79 CYP11B2 (0.40) BACE1KCNH2
SCHEMBL8796991 0.77 POLB (0.40) KCNH2
SCHEMBL8798430 0.75 IMPDH2 (0.43) HTR6CYP2C9LMNACYP1A2PKM
SCHEMBL9088314 0.73 RARA (0.39) HTR6NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514942-B1 Novel benzopyran derivatives and processes for the preparation thereof KOREA RES INST CHEM TECH (KR) 1997-03-05 EP disclosed
US-5493029-A USEFUL IN TREATING ASTHMA AND HYPERTENSION KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1996-02-20 US disclosed
US-5300511-A Spiro-benzopyran derivatives and useful for treating asthma and hypertension KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1994-04-05 US disclosed
EP-0514942-A1 Novel benzopyran derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1992-11-25 EP disclosed