SCHEMBL8801256

SCHEMBL8801256

COc1cc(OC)nc(C2(O)OC(=O)c3cccnc32)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.35
HCRTR2 O43614 3/20 0.35
ADORA2A P29274 1/20 0.33
ELANE P08246 1/20 0.33
CES2 O00748 2/20 0.33
S100A4 P26447 1/20 0.33
HKDC1 Q2TB90 1/20 0.33
PADI1 Q9ULC6 1/20 0.33
PADI3 Q9ULW8 1/20 0.33
PADI4 Q9UM07 1/20 0.33
PADI2 Q9Y2J8 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
NPY5R Q15761 1/20 0.32
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32
BTK Q06187 1/20 0.32
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
IDO1 P14902 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322076 0.79 HCRTR1 (0.36) HCRTR1HCRTR2CES2BTKEDNRB
SCHEMBL8324080 0.77 TUBB4A (0.35) ADORA2ACES2
SCHEMBL8321836 0.76 EDNRA (0.37) CES2EDNRBEDNRACYP1A2CYP2C9
SCHEMBL8319030 0.76 MAOB (0.38) HCRTR1HCRTR2ADORA2A
SCHEMBL8918214 0.75 CES2 (0.36) HCRTR1HCRTR2CES2EDNRBEDNRA
SCHEMBL8576515 0.72 EDNRB (0.33) EDNRBEDNRA
SCHEMBL8572771 0.69 EDNRB (0.34) EDNRBEDNRA
SCHEMBL8693898 0.68 HCAR3 (0.38) CYP1A2CYP2C9CYP2C19TDP2
SCHEMBL8810384 0.68 NPSR1 (0.36) EDNRBEDNRA
SCHEMBL8809785 0.67 HKDC1 (0.35) S100A4HKDC1PADI1PADI3PADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752424-A1 NICOTINIC ACID DERIVATIVE AND HERBICIDE KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1997-01-08 EP disclosed