SCHEMBL8801355

SCHEMBL8801355

CCOC(=O)CN1C(=O)C(NCC(=O)OC(C)(C)C)C=C(c2ccccc2Cl)c2cc(Cl)ccc21

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
CCKBR P32239 8/20 0.42
CCKAR P32238 3/20 0.41
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.37
BRD4 O60885 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801216 0.91 CCKBR (0.39) MAPTCCKBRCCKARUSP2BRD4
SCHEMBL8804138 0.83 CCKBR (0.42) CCKBRCCKAR
SCHEMBL8801767 0.82 BRD4 (0.41) MAPTCCKBRALDH1A1BRD4
SCHEMBL8801349 0.82 HTT (0.45) HTTMAPTTSHRCCKBRCCKAR
SCHEMBL8801124 0.82 CCKBR (0.51) HTTMAPTTSHRCCKBRCCKAR
SCHEMBL8803196 0.74 CCKBR (0.47) CCKBRCCKAR
SCHEMBL8801220 0.72 ALOX15 (0.40) MAPTCCKBRCCKARUSP2BRD4
SCHEMBL8800433 0.71 CCKBR (0.46) CCKBRCCKAR
SCHEMBL9039585 0.68 CCKBR (0.61) CCKBR
SCHEMBL8667990 0.68 CCKBR (0.55) CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0763537-A2 Non-peptidyl Ras farnesyl transferase inhibitors GENENTECH, INC. (US) 1997-03-19 EP disclosed
EP-0698015-A1 PREPARATION OF N-CYANODITHIOIMINO-CARBONATES AND 3-MERCAPTO-5-AMINO-1H-1,2,4-TRIAZOLE GENENTECH, INC. (US) 1996-02-28 EP disclosed
WO-1994026723-A2 ras FARNESYL TRANSFERASE INHIBITORS GENENTECH, INC. (US) 1994-11-24 WO disclosed