SCHEMBL8801767

SCHEMBL8801767

CC(C)(C)OC(=O)CNC1C=C(c2ccccc2)c2cc(Cl)ccc2N(CC(=O)O)C1=O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.41
CCKBR P32239 4/20 0.40
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HDAC3 O15379 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
LMNA P02545 1/20 0.37
OPRK1 P41145 1/20 0.37
PDE3A Q14432 1/20 0.37
CYP1A2 P05177 1/20 0.36
HTR2B P41595 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801216 0.91 CCKBR (0.39) BRD4CCKBRALOX15HSD17B10OPRK1
SCHEMBL8804138 0.90 CCKBR (0.42) CCKBRALOX15HSD17B10OPRK1TP53
SCHEMBL8801355 0.82 HTT (0.43) BRD4CCKBRALDH1A1MAPT
SCHEMBL8667990 0.82 CCKBR (0.55) CCKBRLMNAOPRK1PDE3AHTR2B
SCHEMBL8801763 0.80 ALOX15 (0.41) BRD4CCKBRALOX15HSD17B10LMNA
SCHEMBL8800433 0.78 CCKBR (0.46) CCKBRALOX15HSD17B10OPRK1TP53
SCHEMBL8803196 0.77 CCKBR (0.47) CCKBROPRK1CYP1A2PDE4D
SCHEMBL9039585 0.77 CCKBR (0.61) CCKBR
SCHEMBL8669229 0.76 CCKBR (0.57) CCKBRLMNAMAPT
SCHEMBL8669189 0.72 CCKBR (0.58) CCKBRHDAC3HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0763537-A2 Non-peptidyl Ras farnesyl transferase inhibitors GENENTECH, INC. (US) 1997-03-19 EP disclosed
EP-0698015-A1 PREPARATION OF N-CYANODITHIOIMINO-CARBONATES AND 3-MERCAPTO-5-AMINO-1H-1,2,4-TRIAZOLE GENENTECH, INC. (US) 1996-02-28 EP disclosed
WO-1994026723-A2 ras FARNESYL TRANSFERASE INHIBITORS GENENTECH, INC. (US) 1994-11-24 WO disclosed