SCHEMBL8801521

SCHEMBL8801521

CC(=O)Oc1ccc2c(C=O)c(Cc3ccccc3)[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
GAA P10253 2/20 0.51
GLA P06280 1/20 0.51
AHR P35869 4/20 0.47
IMPDH2 P12268 1/20 0.45
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
PARP1 P09874 1/20 0.40
CA2 P00918 1/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8802154 0.85 KDM4E (0.53) KDM4EGAAGLAMTNR1AMTNR1B
SCHEMBL8801343 0.78 KDM4E (0.47) KDM4EAHRIMPDH2MAPTALDH1A1
SCHEMBL4323256 0.76 GSK3B (0.51) AHRIMPDH2MEN1KMT2A
SCHEMBL6592979 0.74 AHR (0.66) KDM4EAHRIMPDH2MTNR1AMTNR1B
SCHEMBL8801366 0.73 CA2 (0.52) KDM4EGAAGLAMTNR1AMTNR1B
SCHEMBL1180269 0.72 KDM4E (0.61) KDM4EGAAGLAAHRMTNR1A
SCHEMBL28239180 0.72 AHR (0.52) AHRMAPTCA2MEN1HPGD
SCHEMBL11304077 0.70 KDM4E (0.50) KDM4EGAAGLAMAPTALDH1A1
SCHEMBL531085 0.70 ELANE (0.61) GAAMAPTMAPK1ALDH1A1KMT2A
SCHEMBL28490003 0.69 MAOA (0.51) AHRMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804416-A1 HETEROCYCLIC COMPOUNDS, USEFUL AS ALLOSTERIC EFFECTORS AT MUSCARINIC RECEPTORS SANKYO COMPANY LIMITED (JP) 1997-11-05 EP disclosed