SCHEMBL8804587

SCHEMBL8804587

CCOC(Cc1ccc2oc(Cc3ccccc3)nc2c1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPARG P37231 13/20 0.51
PPARA Q07869 9/20 0.51
GAA P10253 1/20 0.48
PPARD Q03181 2/20 0.47
LMNA P02545 1/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808210 0.92 PPARA (0.60) PPARGPPARAPPARD
SCHEMBL8805915 0.88 PPARA (0.47) PPARGPPARAGAAPPARD
SCHEMBL8806855 0.85 PPARG (0.63) PPARGPPARAPPARD
SCHEMBL8805213 0.80 FAAH (0.46) GAALMNARAB9ANPC1
SCHEMBL11638476 0.76 GAA (0.71) GAALMNARAB9ANPC1
SCHEMBL11636604 0.75 RAB9A (0.51) GAALMNARAB9ANPC1
SCHEMBL11638633 0.75 MAOA (0.54) GAALMNARAB9ANPC1
SCHEMBL5766871 0.74 LMNA (0.61) GAALMNARAB9ANPC1
SCHEMBL1670312 0.74 PPARA (0.69) PPARGPPARAPPARD
SCHEMBL4993002 0.74 PPARA (0.69) PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533781-B1 3-ARYL-2-HYDROXYPROPIONIC ACID DERIVATIVES AND ANALOGS AS HYPOGLYCEMIC AGENTS PFIZER (US) 1997-02-26 EP disclosed
US-5438074-A 3-aryl-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents PFIZER INC. (US) 1995-08-01 US disclosed
US-5306726-A 3-aryl-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents PFIZER INC. (US) 1994-04-26 US disclosed
US-5232945-A 3-aryl-2-hydroxypropionic acid derivatives and analogs as antihypertensives PFIZER INC. (US) 1993-08-03 US disclosed
EP-0533781-A1 3-ARYL-2-HYDROXYPROPIONIC ACID DERIVATIVES AND ANALOGS AS HYPOGLYCEMIC AGENTS. PFIZER (US) 1993-03-31 EP disclosed
WO-1991019702-A1 3-ARYL-2-HYDROXYPROPIONIC ACID DERIVATIVES AND ANALOGS AS HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1991-12-26 WO disclosed