SCHEMBL8812136

SCHEMBL8812136

Cc1ccc(-c2ccccc2)c(C(=O)Nc2ccc(C(=O)N(C)c3ccc(Cl)cc3O)cc2C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TP53 P04637 2/20 0.46
ALDH1A1 P00352 2/20 0.44
F10 P00742 3/20 0.43
SERPINE1 P05121 2/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
GAA P10253 2/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
TAS1R2 Q8TE23 1/20 0.42
KCNMA1 Q12791 3/20 0.41
MAPT P10636 2/20 0.40
ALOX12 P18054 1/20 0.40
S1PR4 O95977 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7373393 0.90 ALDH1A1 (0.47) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL8813752 0.90 KCNMA1 (0.49) SMN1; SMN2NPC1TP53ALDH1A1F10
SCHEMBL7513968 0.83 RAB9A (0.46) NPC1RAB9ATP53ALDH1A1F10
SCHEMBL8814928 0.83 NPC1 (0.46) SMN1; SMN2NPC1RAB9ATP53PPARG
SCHEMBL8814391 0.80 POLB (0.46) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL7371628 0.80 KCNMA1 (0.48) SMN1; SMN2NPC1RAB9AALDH1A1F10
SCHEMBL8814366 0.79 CYP19A1 (0.44) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL7376165 0.78 AVPR2 (0.48) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL8816300 0.78 BRD4 (0.45) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL8812151 0.78 GAA (0.41) SMN1; SMN2TP53ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757670-A1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed