SCHEMBL8828099

SCHEMBL8828099

COc1nc2cc(Cl)cc(Cl)c2cc1C[PH](=O)O

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.32
PDCD1LG2 Q9BQ51 2/20 0.32
CD274 Q9NZQ7 2/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828092 0.72 MMP1 (0.36) KMT2AMEN1ALDH1A1HPGD
SCHEMBL8637396 0.72 PTGES (0.36)
SCHEMBL8828082 0.65 GRIN1 (0.45) ALDH1A1
SCHEMBL8612392 0.61 NR4A2 (0.33) ALDH1A1
SCHEMBL8872967 0.59 TSHR (0.40) KMT2AMEN1ALDH1A1HPGD
SCHEMBL5973965 0.59 HRH4 (0.33) KMT2APDCD1LG2CD274MEN1
SCHEMBL7675179 0.59 HRH4 (0.56) KMT2AMEN1
SCHEMBL17372703 0.59 GLP1R (0.48) CYP1A2ALDH1A1HPGDNPSR1
SCHEMBL8071245 0.58 CRHR1 (0.35) ALDH1A1
SCHEMBL8078338 0.58 PDE4A (0.37) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646132-A TREATING CEREBRAL ISCHEMIA ADIR ET COMPAGNIE (FR) 1997-07-08 US disclosed
US-5536709-A INHIBITORS OF HYPERACTIVATION OF EXCITATORY AMINO ACIDS ADIR ET COMPAGNIE (FR) 1996-07-16 US disclosed