SCHEMBL8828347

SCHEMBL8828347

COc1ccc(CCN(C)CCC(C)NC(=O)C/C=C/c2ccc(-n3ccnc3)cc2)cc1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
CYP3A4 P08684 6/20 0.39
CYP2D6 P10635 2/20 0.39
CYP1A2 P05177 1/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
MAPT P10636 2/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
MAOB P27338 1/20 0.39
KDM4E B2RXH2 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH1A1 P00352 5/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
CYP24A1 Q07973 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828534 0.89 CYP24A1 (0.41) POLBCYP2D6CYP1A2MEN1KMT2A
SCHEMBL8828195 0.86 OPRM1 (0.44) CYP3A4CYP2D6CYP1A2MEN1KMT2A
SCHEMBL8828270 0.86 ALDH1A1 (0.39) POLBCYP3A4CYP2D6CYP1A2MEN1
SCHEMBL9233122 0.85 OPRM1 (0.42) CYP3A4CYP2D6CYP1A2MEN1KMT2A
SCHEMBL8828201 0.84 NOS2 (0.40) POLBCYP3A4MEN1KMT2ACYP2C9
SCHEMBL8828232 0.83 ALDH1A1 (0.42) CYP3A4CYP2D6CYP1A2MEN1KMT2A
SCHEMBL9160192 0.80 CYP3A4 (0.38) POLBCYP3A4MEN1KMT2AMAPT
SCHEMBL9160628 0.79 MAOB (0.38) MAOB
SCHEMBL8828419 0.79 MAOB (0.38) MEN1KMT2AMAOBKDM4EALDH1A1
SCHEMBL8828231 0.78 OPRM1 (0.44) CYP3A4CYP2D6CYP1A2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650270-A DETECTABLE SIGNALS FOR LABELS AND ANALYZING NORTHEASTERN UNIVERSITY (US) 1997-07-22 US disclosed
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed
US-4016150-A Sulfur and nitrogen-containing organic compositions processes for making them and fuels and additives containing them THE LUBRIZOL CORPORATION (US) 1977-04-05 US disclosed