SCHEMBL8828516

SCHEMBL8828516

O=C1NC(=O)c2c(CCCN3CCN(c4ccccc4F)CC3)cccc21

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.51
DRD3 P35462 1/20 0.51
HTR1A P08908 6/20 0.51
HTR7 P34969 5/20 0.51
HTR2A P28223 2/20 0.51
HTR6 P50406 2/20 0.51
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
DAO P14920 1/20 0.46
CACNA1G O43497 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7986154 0.84 HTR1A (0.53) DRD2DRD3HTR1AHTR7
SCHEMBL7983420 0.81 HTR1A (0.55) DRD2DRD3HTR1AHTR7
SCHEMBL30080754 0.81 DRD2 (0.60) DRD2DRD3HTR1AHTR7HTR2A
SCHEMBL7986389 0.80 CCR3 (0.50) ADRA1DADRA1AADRA1BKDM4EALDH1A1
SCHEMBL23142609 0.77 CCNE2 (0.43)
SCHEMBL3174237 0.77 CHEK1 (0.47) DRD2DRD3HTR2A
SCHEMBL8557009 0.77 CHEK1 (0.47) HTR2A
SCHEMBL7986525 0.76 CCR3 (0.56) ADRA1DADRA1AADRA1B
SCHEMBL7989675 0.76 SIGMAR1 (0.54) DRD2HTR7TSHR
SCHEMBL8554507 0.76 SIGMAR1 (0.47) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
CN-1136039-A [3- (4-phenylpiperazin-1-yl) propylamino, thio and oxy ] -pyridine, pyrimidine and benzene derivatives HOFFMANN LA ROCHE (CH) 1996-11-20 CN disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed