SCHEMBL883122

SCHEMBL883122

Nc1ccc(CNC(=O)Nc2ccc(C3=NC(c4ccsc4)C(C(=O)NC4CC4)S3)cc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 9/20 0.43
HDAC1 Q13547 4/20 0.41
KLKB1 P03952 1/20 0.34
KDR P35968 2/20 0.33
ROCK2 O75116 2/20 0.33
EPHX1 P07099 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874757 0.75 HDAC1 (0.44) NAMPTHDAC1KLKB1ROCK2
SCHEMBL3050217 0.67 HDAC1 (0.47) NAMPTHDAC1ROCK2
SCHEMBL875591 0.67 NAMPT (0.46) NAMPTHDAC1KLKB1
SCHEMBL3048802 0.66 NAMPT (0.52) NAMPTHDAC1ROCK2
SCHEMBL875577 0.66 HDAC1 (0.43) NAMPTHDAC1KLKB1EPHX1
SCHEMBL15030902 0.66 NPC1 (0.68) NAMPTHDAC1
SCHEMBL875402 0.66 NAMPT (0.45) NAMPTHDAC1KLKB1ROCK2
SCHEMBL3042675 0.66 NAMPT (0.45) NAMPTHDAC1EPHX1
SCHEMBL3045603 0.65 NAMPT (0.50) NAMPTHDAC1
SCHEMBL882752 0.64 NAMPT (0.46) NAMPTHDAC1KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed