SCHEMBL884275

SCHEMBL884275

CC(C)OCCOc1cccc(Cn2c(C(=O)N3CCNCC3)c(-c3ccccc3)n(C3CCCN(C(=O)CI)C3)c2=O)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
PTGIR P43119 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
REN P00797 2/20 0.32
MEN1 O00255 1/20 0.32
ITGB3 P05106 4/20 0.32
ITGA2B P08514 4/20 0.32
POLB P06746 2/20 0.32
USP2 O75604 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2062724 0.93 PTGIR (0.34) ALDH1A1TSHRPTGIRKMT2AMAPT
SCHEMBL884926 0.89 ALDH1A1 (0.44) ALDH1A1TSHRKMT2ANPC1MAPT
SCHEMBL884303 0.89 KDM4E (0.36) ALDH1A1TSHRPTGIRKMT2AMAPT
SCHEMBL885548 0.87 BCL9 (0.36) ALDH1A1KMT2ATP53RENMEN1
SCHEMBL884402 0.87 PTGIR (0.36) ALDH1A1TSHRPTGIRKMT2AMAPT
SCHEMBL884549 0.85 REN (0.39) ALDH1A1TSHRPTGIRKMT2AMAPT
SCHEMBL886063 0.85 ALDH1A1 (0.35) ALDH1A1TSHRPTGIRKMT2ATP53
SCHEMBL885904 0.83 HTR1A (0.36) ALDH1A1TSHRPTGIRKMT2ANPC1
SCHEMBL2062941 0.83 KDM4E (0.38) ALDH1A1TSHRPTGIRKMT2AMAPT
SCHEMBL884381 0.82 KMT2A (0.39) ALDH1A1TSHRPTGIRKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089005-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-07-24 WO claimed
WO-2008089005-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-07-24 WO disclosed