SCHEMBL8865242

SCHEMBL8865242

COc1cc2c(cc1OC)C(c1c[nH]cn1)CCC2

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.41
MAOA P21397 3/20 0.40
TSHR P16473 1/20 0.40
ABCB1 P08183 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
KMT2A Q03164 1/20 0.38
EP300 Q09472 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865285 0.82 GID4 (0.50) CHRNA7
SCHEMBL8865311 0.80 ALOX15 (0.51) TSHRCYP3A4CYP2D6
SCHEMBL8865945 0.80 HTR1A (0.41)
Hydrochloric Acid SCHEMBL8865276 0.78 ALOX15 (0.50) TSHRCYP3A4CYP2D6
SCHEMBL8865236 0.78 ADRA1A (0.51) CA1CA2
SCHEMBL8865117 0.77 SRD5A1 (0.39) CYP3A4CYP2D6KMT2A
SCHEMBL8865462 0.76 PARP1 (0.43) MAOACA1CA2
SCHEMBL7604210 0.75 ADRA1A (0.38) KMT2A
SCHEMBL7097683 0.75 ADRA1A (0.40) CA1CA2
SCHEMBL7607644 0.75 CYP19A1 (0.46) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US claimed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP claimed
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US disclosed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP disclosed