SCHEMBL8872029

SCHEMBL8872029

CCCCN(c1ccncc1N)N1C(=O)C(C)c2ccccc21

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.33
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CNR2 P34972 3/20 0.32
CNR1 P21554 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
TP53 P04637 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8872220 0.72 LMNA (0.31) ALDH1A1LMNA
SCHEMBL8872371 0.72 SLC6A2 (0.31) SLC6A2
SCHEMBL9198258 0.71 KMT2A (0.31) SLC6A2KMT2A
SCHEMBL9379716 0.68 CYP19A1 (0.32) SLC6A2KMT2A
SCHEMBL8872591 0.67 CES2 (0.34) SLC6A2ALDH1A1MEN1KMT2A
SCHEMBL8860275 0.66 ALDH1A1 (0.31) ALDH1A1
SCHEMBL8871301 0.66 LMNA (0.31) ALDH1A1LMNA
SCHEMBL26056119 0.66 AOC1 (0.38) SLC6A2ALDH1A1MEN1KMT2AMAPT
SCHEMBL8872035 0.65 AOC1 (0.33) LMNA
SCHEMBL9206194 0.62 SLC6A2 (0.34) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5621116-A CHEMICAL INTERMEDIATES; MEMORY ENHANCERS FOR TREATMENT OF ALZHEIMER*S, ANALGESICS, ANTICONVULSANTS HOECHST MARION ROUSSEL, INC. (US) 1997-04-15 US disclosed
EP-0415102-B1 1,3-Dihydro-1-(pyridinylamino)-2H-indol-2-ones, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1995-02-01 EP disclosed
US-5179119-A Cognition activators; alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-12 US disclosed
US-5053511-A Analgesics; anticonvulsants; treatment for alzheimers disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-10-01 US disclosed
US-5006537-A Analgesics, memory enhancement, Alzheimer* disease HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-04-09 US disclosed
EP-0415102-A1 1,3-Dihydro-1-(pyridinylamino)-2H-indol-2-ones, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-03-06 EP disclosed