SCHEMBL8875707

SCHEMBL8875707

CC1(C(=O)O)C(=O)c2cc(C#N)ccc2OC1c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 5/20 0.36
ABCB1 P08183 6/20 0.36
DNMT3B Q9UBC3 1/20 0.36
CXCR2 P25025 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
KDM4E B2RXH2 1/20 0.35
PTGS2 P35354 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25201529 0.81 DNMT3B (0.52) DNMT3BCYP3A4KDM4E
Hydrochloric Acid SCHEMBL11091455 0.70 MEN1 (0.46) ABCB1DNMT3BCYP3A4KDM4E
SCHEMBL7269358 0.64 PBRM1 (0.61) ABCB1PTGS2
SCHEMBL2471424 0.63 MALT1 (0.43) ABCC9ABCB1CYP3A4KDM4E
SCHEMBL9819081 0.63 SIGMAR1 (0.46) ABCB1KDM4E
SCHEMBL31103518 0.62 NOS3 (0.44) ALOX15PTGDR2
SCHEMBL3518800 0.62 ALDH1A1 (0.36) DNMT3BKDM4E
SCHEMBL5313705 0.61 DNMT3B (0.57) DNMT3BCYP3A4KDM4E
SCHEMBL11574836 0.61 DNMT3B (0.39) ABCB1DNMT3BKDM4EPTGS2
SCHEMBL11572960 0.61 DNMT3B (0.44) ABCB1DNMT3BKDM4EPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US disclosed
US-5474994-A Treating hypertension, urethral and lower urinary tract contractions RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-12-12 US disclosed