SCHEMBL8888264

SCHEMBL8888264

CC(C)Oc1cccc(-c2n[nH]c(-c3ccccc3)c2-c2ccc(=O)[nH]n2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
GABRA1 P14867 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
PDE3A Q14432 4/20 0.38
PDE5A O76074 1/20 0.38
GPR119 Q8TDV5 1/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 2/20 0.37
CCNE2 O96020 2/20 0.37
CDK4 P11802 2/20 0.37
CCND1 P24385 2/20 0.37
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
DHODH Q02127 1/20 0.37
NR1H2 P55055 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8886941 0.88 NR1H2 (0.49) CYP1A2LMNATP53CCNE2CDK4
SCHEMBL8888641 0.85 MAPT (0.46) CYP1A2RXRARXRBTP53MEN1
SCHEMBL8889732 0.82 CYP1A2 (0.41) CYP1A2GPR119LMNATP53CCNE2
SCHEMBL8887621 0.82 CYP1A2 (0.50) CYP1A2GPR119LMNATP53CCNE2
SCHEMBL8889202 0.80 CYP1A2 (0.41) CYP1A2GPR119TP53MEN1KMT2A
SCHEMBL8890194 0.79 CYP1A2 (0.50) CYP1A2GPR119CCNE2CDK4CCND1
SCHEMBL8887885 0.79 CYP1A2 (0.50) CYP1A2GPR119LMNATP53MAPK1
SCHEMBL8888361 0.79 CYP1A2 (0.50) CYP1A2GPR119TP53HPGDMAPT
SCHEMBL8889663 0.79 CYP1A2 (0.47) CYP1A2PDE3APDE5AGPR119LMNA
SCHEMBL8889051 0.78 LMNA (0.60) CYP1A2LMNATP53CCNE2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed