SCHEMBL8898526

SCHEMBL8898526

COCCNc1nc(NCC2CCC(CN)CC2)nc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.50
CYP3A4 P08684 9/20 0.50
HSD17B10 Q99714 4/20 0.50
USP2 O75604 4/20 0.50
CLK4 Q9HAZ1 3/20 0.50
PDE5A O76074 1/20 0.49
KDM4E B2RXH2 2/20 0.49
CYP2C19 P33261 4/20 0.48
CYP2D6 P10635 4/20 0.48
ALDH1A1 P00352 2/20 0.48
ALOX15 P16050 2/20 0.48
MAPK1 P28482 1/20 0.48
LDHA P00338 1/20 0.47
TSHR P16473 4/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889084 0.94 CASP6 (0.50) CYP1A2CYP3A4HSD17B10USP2CLK4
SCHEMBL8898278 0.88 SOS1 (0.52) PDE5AKDM4EALDH1A1KMT2ALMNA
SCHEMBL8898351 0.87 VCP (0.48) CYP1A2CYP3A4HSD17B10USP2CLK4
SCHEMBL8901747 0.85 TAAR1 (0.56) USP2KDM4EALDH1A1MAPK1TSHR
SCHEMBL8898947 0.85 TLR9 (0.51) PDE5AALDH1A1MAPK1APPCASP6
SCHEMBL8889922 0.84 NPY5R (0.49) PDE5AALDH1A1MAPTHPGDTDP1
SCHEMBL13796628 0.84 NPY5R (0.55) CYP1A2CYP3A4HSD17B10USP2CLK4
SCHEMBL8898707 0.83 FLT3 (0.48) APPCASP6TLR7SOS1TRIM58
SCHEMBL8907323 0.83 TRIM58 (0.57) ALDH1A1MAPK1KMT2ACASP6TRIM58
SCHEMBL8899155 0.83 TRIM58 (0.57) ALDH1A1MAPK1KMT2ACASP6TRIM58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020823-A2 2-AMINO QUINAZOLINE DERIVATIVES AS NPY RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 1997-06-12 WO disclosed