SCHEMBL889285

SCHEMBL889285

Nc1ncnc2c1ccn2C1CC(O)C(COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.58
TRPM2 O94759 1/20 0.54
METTL3 Q86U44 3/20 0.53
PRMT5 O14744 2/20 0.53
P2RY1 P47900 4/20 0.53
ENPP1 P22413 2/20 0.53
P2RX1 P51575 2/20 0.52
P2RX3 P56373 2/20 0.52
P2RX2 Q9UBL9 2/20 0.52
DTYMK P23919 2/20 0.51
P2RY2 P41231 4/20 0.51
P2RY4 P51582 2/20 0.51
P2RY6 Q15077 2/20 0.51
SRC P12931 1/20 0.49
P2RX4 Q99571 1/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
RNASEL Q05823 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29487848 1.00 POLB (0.58) POLBTRPM2METTL3PRMT5P2RY1
SCHEMBL26031206 1.00 POLB (0.58) POLBTRPM2METTL3PRMT5P2RY1
SCHEMBL16743500 0.89 POLB (0.63) POLBTRPM2P2RY1ENPP1P2RX1
SCHEMBL16743926 0.89 POLB (0.63) POLBTRPM2P2RY1ENPP1P2RX1
SCHEMBL18520880 0.88 METTL3 (0.57) POLBTRPM2METTL3PRMT5P2RY1
SCHEMBL27337818 0.85 P2RX3 (0.45) POLBP2RY1P2RX1P2RX3P2RX2
SCHEMBL5044161 0.84 POLB (0.80) POLBTRPM2P2RY1ENPP1P2RX1
SCHEMBL889289 0.84 POLB (0.80) POLBTRPM2P2RY1ENPP1P2RX1
SCHEMBL14471000 0.84 POLB (0.80) POLBTRPM2P2RY1ENPP1P2RX1
Tubercidin Triphosphate SCHEMBL12932266 0.84 P2RY1 (0.67) TRPM2P2RY1P2RX1P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170275672-A1 CHEMICALLY MODIFIED LIGASE COFACTORS, DONORS AND ACCEPTORS TRILINK BIOTECHNOLOGIES, INC. (US) 2017-09-28 US disclosed
US-20170275672-A1 CHEMICALLY MODIFIED LIGASE COFACTORS, DONORS AND ACCEPTORS TRILINK BIOTECHNOLOGIES, INC. (US) 2017-09-28 US disclosed
US-9631227-B2 Chemically modified ligase cofactors, donors and acceptors TRILINK BIOTECHNOLOGIES, INC. (US) 2017-04-25 US disclosed
US-9631227-B2 Chemically modified ligase cofactors, donors and acceptors TRILINK BIOTECHNOLOGIES, INC. (US) 2017-04-25 US disclosed
US-20140323354-A1 Chemically Modified Ligase Cofactors, Donors and Acceptors TRILINK BIOTECHNOLOGIES, INC. (US) 2014-10-30 US disclosed
US-20140323354-A1 Chemically Modified Ligase Cofactors, Donors and Acceptors TRILINK BIOTECHNOLOGIES, INC. (US) 2014-10-30 US disclosed
WO-2014144979-A1 CHEMICALLY MODIFIED LIGASE COFACTORS, DONORS AND ACCEPTORS TRILINK BIOTECHNOLOGIES, INC. (US) 2014-09-18 WO disclosed
US-8728725-B2 Chemically modified ligase cofactors, donors and acceptors TRILINK BIOTECHNOLOGIES (US) 2014-05-20 US disclosed
US-8728725-B2 Chemically modified ligase cofactors, donors and acceptors TRILINK BIOTECHNOLOGIES (US) 2014-05-20 US disclosed
US-20110045485-A1 ANALYTICAL METHOD AND KIT ENIGMA DIAGNOSTICS LIMITED (GB) 2011-02-24 US disclosed
US-20110008788-A1 CHEMICALLY MODIFIED LIGASE COFACTORS, DONORS AND ACCEPTORS TriLink Bio Technologies 2011-01-13 US disclosed
US-20110008788-A1 CHEMICALLY MODIFIED LIGASE COFACTORS, DONORS AND ACCEPTORS TriLink Bio Technologies 2011-01-13 US disclosed
WO-2011005762-A1 CHEMICALLY MODIFIED LIGASE COFACTORS, DONORS AND ACCEPTORS TRILINK BIOTECHNOLOGIES (US) 2011-01-13 WO disclosed
US-7838236-B2 Analytical method and kit ENIGMA DIAGNOSTICS LIMITED (GB) 2010-11-23 US disclosed
US-7838236-B2 Analytical method and kit ENIGMA DIAGNOSTICS LIMITED (GB) 2010-11-23 US disclosed
US-20080233588-A1 Analytical Method and Kit ENIGMA DIAGNOSTICS LIMITED (GB) 2008-09-25 US disclosed
US-20080233588-A1 Analytical Method and Kit ENIGMA DIAGNOSTICS LIMITED (GB) 2008-09-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110045485-A1 ANALYTICAL METHOD AND KIT RNGTT, ADAR, RNASE1 POLB 95/4885TRPM2 4276/4885METTL3 305/4885
US-20080233588-A1 Analytical Method and Kit RNGTT, ADAR, RNASE1 POLB 69/4885TRPM2 4201/4885METTL3 516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.