SCHEMBL8892874

SCHEMBL8892874

CCOc1ccc(CC(=O)NC(CC)c2ccsc2)cc1S(=O)(=O)NC(=O)NC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 2/20 0.36
SLC22A1 O15245 1/20 0.36
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36
NR1I2 O75469 1/20 0.36
ABCB11 O95342 1/20 0.36
LMNA P02545 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
HTR2A P28223 1/20 0.36
MAPK1 P28482 1/20 0.36
ADRA1A P35348 1/20 0.36
PTGS2 P35354 1/20 0.36
PDE4D Q08499 1/20 0.36
ABCC8 Q09428 1/20 0.36
NR1I3 Q14994 1/20 0.36
ABCC2 Q92887 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
PTPRB P23467 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890891 0.93 KEAP1 (0.37) ALDH1A1LMNAPTPRBTBXA2RMAPT
SCHEMBL8891439 0.92 PTPRB (0.40) POLBLMNAMAPK1ABCC8PTPRB
SCHEMBL8890922 0.91 ABCC8 (0.38) ALDH1A1POLBCYP3A4SLC22A1ABCC3
SCHEMBL8893995 0.91 ALDH1A1 (0.41) ALDH1A1POLBCYP3A4SLC22A1ABCC3
SCHEMBL8892721 0.87 IDH1 (0.35) ALDH1A1POLBLMNAPTPRBSMN1; SMN2
SCHEMBL8892008 0.85 PTPRB (0.31) PTPRB
SCHEMBL8892165 0.85 ABCC9 (0.37) ALDH1A1LMNAABCC8PTPRBTBXA2R
SCHEMBL8893620 0.84 ALDH1A1 (0.34) ALDH1A1POLBCYP3A4SLC22A1ABCC3
SCHEMBL8893013 0.84 ALDH1A1 (0.34) ALDH1A1POLBCYP3A4SLC22A1ABCC3
SCHEMBL8892364 0.84 KEAP1 (0.38) ALDH1A1POLBTBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607976-A ANNTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-03-04 US disclosed