SCHEMBL8893501

SCHEMBL8893501

CCCN1CN(CC(=O)OC)C(=O)C12CCN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 3/20 0.53
NPC1L1 Q9UHC9 8/20 0.43
OPRL1 P41146 2/20 0.38
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 1/20 0.37
DDR1 Q08345 3/20 0.36
CCR5 P51681 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8892471 0.89 BDKRB2 (0.55) BDKRB2NPC1L1OPRM1OPRK1DDR1
SCHEMBL8910702 0.84 BDKRB2 (0.52) BDKRB2NPC1L1OPRL1OPRM1OPRK1
SCHEMBL8892630 0.79 NPC1L1 (0.67) BDKRB2NPC1L1OPRL1OPRM1OPRK1
SCHEMBL8893884 0.78 NPC1L1 (0.56) BDKRB2NPC1L1OPRL1OPRM1OPRK1
SCHEMBL8894056 0.75 BDKRB2 (0.59) BDKRB2NPC1L1
SCHEMBL21068971 0.75 CYP2D6 (0.50) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL8893424 0.74 CCR5 (0.51) NPC1L1OPRM1OPRK1CCR5
SCHEMBL599707 0.73 NAMPT (0.39)
SCHEMBL5134369 0.73 GRIN2B (0.47) BDKRB2NPC1L1OPRL1OPRM1OPRK1
SCHEMBL4130653 0.72 CCR5 (0.39) NPC1L1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610142-A Bradykinin antagonist pseudopeptide derivatives of substituted 4-keto-1,3,8-triazaspiro[4.5]decan-3-alkanoic acids SCIOS INC. (US) 1997-03-11 US disclosed