SCHEMBL8900865

SCHEMBL8900865

COC(=O)CC1C(=O)CCc2c(OC)cccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.43
TAS1R1 Q7RTX1 2/20 0.43
TAS1R2 Q8TE23 2/20 0.43
POLL Q9UGP5 1/20 0.43
KMT2A Q03164 2/20 0.43
GAA P10253 1/20 0.43
EGFR P00533 1/20 0.41
HTR2A P28223 1/20 0.41
MAPT P10636 2/20 0.41
CYP1A2 P05177 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9441289 0.89 CYP1A2 (0.43) TAS1R3TAS1R1TAS1R2POLLKMT2A
SCHEMBL8900041 0.79 HTR1A (0.43) KMT2AGAAHTR2AMAPTCYP1A2
SCHEMBL8168722 0.78 EGFR (0.48) KMT2AGAAEGFRHTR2AMAPT
SCHEMBL7926481 0.77 HTR1A (0.46) POLLKMT2AHTR2ACYP1A2MEN1
SCHEMBL11978323 0.75 KDM4E (0.41) KMT2AGAAMAPTCYP1A2CA1
SCHEMBL9309831 0.74 ACHE (0.49) POLLKMT2AGAACYP1A2CA1
SCHEMBL9441282 0.73 MTNR1A (0.44) TAS1R3TAS1R1TAS1R2POLLKMT2A
SCHEMBL24650908 0.71 DRD2 (0.42) MAPTCYP1A2CA1CA2DRD2
SCHEMBL11957274 0.71 CYP1A2 (0.38) KMT2AGAAMAPTCYP1A2CA1
SCHEMBL11363652 0.70 CYP1A2 (0.48) POLLKMT2AGAAEGFRHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482084-B1 (1,2N) AND (3,2N)-CARBOCYCLIC-2-AMINO TETRALIN DERIVATIVES UPJOHN CO (US) 1997-05-07 EP disclosed
US-5491236-A NERVOUS SYTEM DISORDERS THE UPJOHN COMPANY (US) 1996-02-13 US disclosed