SCHEMBL8900041

SCHEMBL8900041

COC(=O)CC1C(=O)CCc2cccc(OC)c21

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.43
GAA P10253 1/20 0.43
KMT2A Q03164 1/20 0.43
MTNR1B P49286 9/20 0.41
MTNR1A P48039 8/20 0.41
HTR2A P28223 1/20 0.41
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9372184 0.88 HTR2A (0.42) HTR1AMTNR1BMTNR1AHTR2ACYP2D6
SCHEMBL8900865 0.79 TAS1R3 (0.43) HTR1AGAAKMT2AMTNR1BMTNR1A
SCHEMBL7926754 0.78 HTR1A (0.55) HTR1AHTR2A
SCHEMBL7935755 0.78 HTR1A (0.52) HTR1AKMT2AMTNR1BMTNR1ACYP1A2
SCHEMBL8168722 0.78 EGFR (0.48) GAAKMT2AHTR2ACYP2D6CYP1A2
SCHEMBL7926523 0.77 HTR1A (0.53) HTR1AHTR2A
SCHEMBL7935873 0.76 MTNR1A (0.43) HTR1AKMT2AMTNR1BMTNR1ACYP2D6
SCHEMBL9052842 0.74 DRD2 (0.45) HTR1A
SCHEMBL9441175 0.73 MTNR1B (0.44) HTR1AMTNR1BMTNR1AHTR2A
SCHEMBL10394822 0.73 MTNR1B (0.51) HTR1AMTNR1BMTNR1ACYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482084-B1 (1,2N) AND (3,2N)-CARBOCYCLIC-2-AMINO TETRALIN DERIVATIVES UPJOHN CO (US) 1997-05-07 EP disclosed
US-5491236-A NERVOUS SYTEM DISORDERS THE UPJOHN COMPANY (US) 1996-02-13 US disclosed