SCHEMBL8904626

SCHEMBL8904626

CSc1ccc(C(=O)c2ccc(C(C)c3ccc(=O)[nH]n3)[nH]2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
TSHR P16473 1/20 0.48
NFKB1 P19838 1/20 0.48
PDE4A P27815 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
ATM Q13315 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PLK1 P53350 1/20 0.32
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8904899 0.88 GRK6 (0.35) CYP1A2CYP3A4CYP2C9HPGDALOX15
SCHEMBL8905805 0.87 LMNA (0.38) CYP1A2CYP3A4CYP2C9HPGDALOX15
SCHEMBL8905900 0.86 LMNA (0.37) CYP1A2CYP3A4CYP2C9HPGDTSHR
SCHEMBL8904194 0.86 CCNA2 (0.38) CYP1A2CYP3A4CYP2C9HPGDALOX15
SCHEMBL8906156 0.86 ALDH1A1 (0.35) CYP2C9HPGDMEN1KMT2A
SCHEMBL8905938 0.86 MEN1 (0.38) CYP1A2CYP3A4CYP2C9HPGDALOX15
SCHEMBL9030270 0.85 PDE3B (0.42) CYP1A2CYP3A4HPGDPDE4APDE4B
SCHEMBL8904850 0.85 ALDH1A1 (0.40) CYP1A2CYP3A4CYP2C9HPGDTSHR
SCHEMBL8904827 0.84 PDE3B (0.36) CYP1A2HPGDPDE4APDE4BPDE4C
SCHEMBL8904574 0.84 NPC1 (0.42) HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622948-A ANALGESICS SYNTEX (U.S.A.) INC. (US) 1997-04-22 US disclosed
EP-0714895-A1 Pyrrole derivatives F. Hoffmann-La Roche AG (CH) 1996-06-05 EP disclosed