SCHEMBL8905938

SCHEMBL8905938

CC(c1ccc(=O)[nH]n1)c1ccc(C(=O)c2ccc(F)cc2)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LTA4H P09960 1/20 0.37
AKR1B1 P15121 2/20 0.35
GRM5 P41594 1/20 0.33
MAPK1 P28482 2/20 0.32
RXFP1 Q9HBX9 2/20 0.32
ADORA3 P0DMS8 1/20 0.32
PTGS1 P23219 1/20 0.32
KDR P35968 1/20 0.32
ALDH1A1 P00352 5/20 0.31
HTT P42858 2/20 0.31
HPGD P15428 2/20 0.31
PDE3B Q13370 2/20 0.31
PDE3A Q14432 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905805 0.89 LMNA (0.38) MEN1KMT2AAKR1B1ALDH1A1HTT
SCHEMBL8906156 0.88 ALDH1A1 (0.35) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL8904194 0.88 CCNA2 (0.38) MEN1KMT2AAKR1B1MAPK1RXFP1
SCHEMBL8905900 0.88 LMNA (0.37) MEN1KMT2AAKR1B1MAPK1ADORA3
SCHEMBL8904850 0.88 ALDH1A1 (0.40) MEN1KMT2AAKR1B1ALDH1A1HTT
SCHEMBL9030270 0.88 PDE3B (0.42) MEN1KMT2ALTA4HALDH1A1HTT
SCHEMBL8905725 0.87 AKR1B1 (0.38) AKR1B1NPC1
SCHEMBL8904574 0.86 NPC1 (0.42) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL8904827 0.86 PDE3B (0.36) MEN1KMT2AALDH1A1HTTHPGD
SCHEMBL8904626 0.86 CYP1A2 (0.48) MEN1KMT2AHPGDPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622948-A ANALGESICS SYNTEX (U.S.A.) INC. (US) 1997-04-22 US disclosed
EP-0714895-A1 Pyrrole derivatives F. Hoffmann-La Roche AG (CH) 1996-06-05 EP disclosed