SCHEMBL8907404

SCHEMBL8907404

Nc1ncnc2c1ncn2CCN1C(=O)CSC1COC(=O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.49
ADORA2A P29274 4/20 0.44
SRC P12931 1/20 0.41
KDR P35968 1/20 0.41
PI4KA P42356 1/20 0.41
PI4K2B Q8TCG2 1/20 0.41
PI4K2A Q9BTU6 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
ADORA1 P30542 1/20 0.41
STING1 Q86WV6 1/20 0.41
ADCY5 O95622 3/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GSK3A P49840 1/20 0.40
RPS6KA3 P51812 1/20 0.40
MAPK14 Q16539 1/20 0.40
ALDH1A1 P00352 1/20 0.39
FGFR1 P11362 1/20 0.39
SLC22A6 Q4U2R8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908017 0.83 ADORA2A (0.54) ADORA2AADORA1ADCY5FGFR1SLC22A6
SCHEMBL8909572 0.77 CHRNB2 (0.36) LMNAALDH1A1FGFR1
SCHEMBL8900287 0.77 EP300 (0.38)
SCHEMBL10836169 0.76 EGFR (0.56) EGFRADORA2ASRCKDRPI4KA
SCHEMBL8908130 0.74 CHRNB2 (0.43) SMN1; SMN2
SCHEMBL9836401 0.74 EGFR (0.56) EGFRADORA2ASRCKDRPI4KA
SCHEMBL9836404 0.74 EGFR (0.56) EGFRADORA2ASRCKDRPI4KA
SCHEMBL8901990 0.72 TK1 (0.52) HPGD
SCHEMBL4094131 0.71 EGFR (0.64) EGFRADORA2ASRCKDRPI4KA
SCHEMBL9836909 0.70 EGFR (0.54) EGFRADORA2ASRCKDRPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997034891-A1 SUBSTITUTED 1,3-THIAZOLIDINES AND 1,3-THIAZOLIDIN-4-ONES, METHOD FOR PREPARING SAME, AND USE THEREOF AS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-09-25 WO claimed
WO-1997034891-A1 SUBSTITUTED 1,3-THIAZOLIDINES AND 1,3-THIAZOLIDIN-4-ONES, METHOD FOR PREPARING SAME, AND USE THEREOF AS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-09-25 WO disclosed