SCHEMBL8910252

SCHEMBL8910252

COc1ccc2[nH]c(C(=O)N(C(Cc3c[nH]cn3)C(N)=O)[C@@H](CC3CCCCC3)[C@@H](O)[C@@H](O)C3CC3)cc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.39
ALDH1A1 P00352 4/20 0.37
HPGD P15428 4/20 0.37
HSD17B10 Q99714 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
FLT3 P36888 1/20 0.36
USP2 O75604 1/20 0.35
AKR1C3 P42330 1/20 0.35
TSHR P16473 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PYGL P06737 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8909458 0.91 PYGL (0.36) KDM4EAKR1C3PYGLNPC1RAB9A
SCHEMBL8909154 0.90 REN (0.41) FLT3PDGFRBPYGLHRH4REN
SCHEMBL8910563 0.89 REN (0.41) KDM4EALDH1A1HPGDHSD17B10FLT3
SCHEMBL8910700 0.88 REN (0.40) KDM4EHSD17B10AKR1C3PYGLREN
SCHEMBL8910523 0.83 KDM4E (0.38) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL8908817 0.80 REN (0.38) REN
SCHEMBL8909363 0.77 P2RX1 (0.52) AKR1C3REN
SCHEMBL8909424 0.74 SIRT2 (0.34) AKR1C3PYGLREN
SCHEMBL8910552 0.73 REN (0.36) REN
SCHEMBL8910197 0.73 REN (0.36) MEN1KMT2APYGLREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688946-A DIPEPTIDES FOR HYPOTENSIVE AGENTS AND CARDIOVASCULAR DISORDERS HOFFMANN LA ROCHE INC. (US) 1997-11-18 US disclosed