SCHEMBL8911745

SCHEMBL8911745

CC1=c2c(cc3c(c2C)-c2cccc(F)c2N=3)N=C1C(=O)OCc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.36
RAB9A P51151 5/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
TDP1 Q9NUW8 2/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP12 P39900 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910413 0.89 FGB (0.41) MAPTSMN1; SMN2LMNAALDH1A1KDM4E
SCHEMBL1388443 0.76 DHODH (0.38) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL7966221 0.74 TDP1 (0.38) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL9434331 0.74 TDP1 (0.36) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL9434825 0.72 DHODH (0.38) MAPTRAB9AALDH1A1GPBAR1CYP1A2
SCHEMBL1388453 0.72 TDP1 (0.35) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL9212581 0.72 DHODH (0.38) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL8363373 0.69 TDP1 (0.38) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL8911173 0.65 TDP1 (0.39) MAPTRAB9ASMN1; SMN2NPC1LMNA
SCHEMBL26773019 0.65 ALDH1A1 (0.59) MAPTRAB9ASMN1; SMN2NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US disclosed
CN-1088209-A Heterogeneous ring compound WELLCOME FOUND (GB) 1994-06-22 CN disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed