SCHEMBL8916801

SCHEMBL8916801

CCC(C)(C)Nc1c(C(=O)OC(C)(C)C)ccnc1N1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HRH4 Q9H3N8 4/20 0.36
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
HTR2C P28335 3/20 0.34
HRH3 Q9Y5N1 1/20 0.34
EPHX2 P34913 1/20 0.34
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916074 0.88 HRH4 (0.39) ATRALDH1A1HRH4ACACBACACA
SCHEMBL8916435 0.84 ATR (0.36) ATRALDH1A1HRH4ACACBACACA
SCHEMBL8915723 0.84 ATR (0.36) ATRALDH1A1HRH4ACACBACACA
SCHEMBL8916060 0.83 PRKD1 (0.40) ATRALDH1A1HRH4ADRA1AADRA1B
SCHEMBL8915788 0.80 HTR2C (0.40) HTR2CHRH3EPHX2
SCHEMBL8917894 0.77 HTR2C (0.38) HRH4ADRA1AADRA1BHTR2CHRH3
SCHEMBL27786900 0.75 ALDH1A1 (0.39) ALDH1A1HTR2CEPHX2
SCHEMBL4826186 0.72 PRKCQ (0.41) ATRHRH4ADRA1AADRA1BHRH3
SCHEMBL4738517 0.69 ADRA1A (0.36) HRH4ACACBACACAADRA1AADRA1B
SCHEMBL8219392 0.67 ADRB1 (0.49) ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed