SCHEMBL8918636

SCHEMBL8918636

O=c1oc2cc(Br)cnc2n1CCc1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
KMO O15229 1/20 0.39
HRH1 P35367 1/20 0.39
HTR6 P50406 1/20 0.39
NPC1 O15118 1/20 0.39
DAO P14920 1/20 0.39
PKM P14618 1/20 0.38
AGTR1 P30556 1/20 0.38
PLK1 P53350 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CACNA1B Q00975 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8919447 0.83 KMO (0.41) HSD17B10ALDH1A1KDM4EKMONPC1
SCHEMBL8919804 0.80 LMNA (0.42) HSD17B10ALDH1A1KDM4ENPC1PKM
SCHEMBL7316292 0.76 NPC1 (0.63) HSD17B10ALDH1A1KDM4ENPC1LMNA
SCHEMBL17418888 0.73 PDE4B (0.43) HSD17B10ALDH1A1KDM4ENPC1PKM
SCHEMBL8918139 0.73 HSD17B10 (0.38) HSD17B10ALDH1A1KMONPC1TSHR
SCHEMBL9646262 0.72 HTR1A (0.54)
SCHEMBL8627148 0.70 PDE4B (0.36) HSD17B10ALDH1A1KDM4EKMONPC1
SCHEMBL7328412 0.70 HSD17B10 (0.53) HSD17B10ALDH1A1KDM4ENPC1PKM
SCHEMBL25865447 0.68 HSD17B10 (0.39) HSD17B10ALDH1A1NPC1LMNATSHR
SCHEMBL11343195 0.68 MIF (0.60) ALDH1A1LMNATSHRMAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed