SCHEMBL8920378

SCHEMBL8920378

CC(=O)NC(C=O)(c1ccccc1)c1ccncc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
JAK2 O60674 1/20 0.42
TYK2 P29597 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
TP53 P04637 2/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
STAT3 P40763 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KCNK3 O14649 1/20 0.39
HSD17B10 Q99714 2/20 0.38
NAPRT Q6XQN6 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
PLOD2 O00469 1/20 0.38
PLOD3 O60568 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920573 0.86 RAB9A (0.49) HTTTAAR1TP53KDM4EPOLB
SCHEMBL8920367 0.84 ALDH1A1 (0.49) HTTROCK2ROCK1SMN1; SMN2ALDH1A1
SCHEMBL20986637 0.76 KCNN4 (0.39) SMN1; SMN2HSD17B10ALDH1A1CYP1A2CYP2C9
SCHEMBL8285639 0.73 MAPT (0.42) HTTPOLBHSD17B10ALDH1A1CYP1A2
SCHEMBL31620694 0.70 KIF11 (0.42) HTTJAK2TYK2TAAR1PLOD2
SCHEMBL8695362 0.69 KIF11 (0.46) HTTJAK2TYK2TAAR1ROCK2
SCHEMBL8226385 0.68 KCNN4 (0.50) TAAR1POLBHSD17B10NAPRTALDH1A1
SCHEMBL3322720 0.68 MAPT (0.50) TAAR1POLBHSD17B10NAPRTALDH1A1
SCHEMBL31358110 0.68 KCNN4 (0.47) TAAR1POLBHSD17B10NAPRTALDH1A1
SCHEMBL11298115 0.68 AKR1C3 (0.42) HTTJAK2TYK2TAAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0727998-A4 OXAZOLES FOR TREATING CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORP (US) 1997-03-19 EP disclosed
EP-0727998-A1 OXAZOLES FOR TREATING CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORPORATION (US) 1996-08-28 EP disclosed
WO-1995013067-A1 OXAZOLES FOR TREATING CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORPORATION (US) 1995-05-18 WO disclosed