SCHEMBL8920367

SCHEMBL8920367

COc1cccc(C(C=O)(NC(C)=O)c2ccncc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
RAF1 P04049 1/20 0.44
CYP2D6 P10635 3/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP1B1 Q16678 1/20 0.43
LMNA P02545 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.43
HTT P42858 2/20 0.43
RAB9A P51151 2/20 0.43
GAA P10253 1/20 0.43
ROCK2 O75116 7/20 0.42
ROCK1 Q13464 5/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
PRKACA P17612 2/20 0.42
GSK3A P49840 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920378 0.84 HTT (0.42) ALDH1A1KMT2ACYP2D6CYP1A2LMNA
SCHEMBL8920573 0.77 RAB9A (0.49) ALDH1A1KMT2AMEN1SMN1; SMN2MAPT
SCHEMBL14519898 0.74 ALDH1A1 (0.51) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL29675690 0.74 ALDH1A1 (0.51) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL6207517 0.68 MAPT (0.44) ALDH1A1CYP1A2LMNASMN1; SMN2MAPT
SCHEMBL3532850 0.67 NPC1 (0.44) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL8523810 0.66 KDM4E (0.45) KMT2AMEN1CYP2D6CYP1A2LMNA
SCHEMBL15286571 0.66 ACHE (0.42) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL29039593 0.66 CES2 (0.50) ALDH1A1LMNASMN1; SMN2MAPTHTT
SCHEMBL16147603 0.66 NPSR1 (0.44) ALDH1A1KMT2AMEN1CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0727998-A4 OXAZOLES FOR TREATING CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORP (US) 1997-03-19 EP disclosed
EP-0727998-A1 OXAZOLES FOR TREATING CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORPORATION (US) 1996-08-28 EP disclosed
WO-1995013067-A1 OXAZOLES FOR TREATING CYTOKINE MEDIATED DISEASES SMITHKLINE BEECHAM CORPORATION (US) 1995-05-18 WO disclosed