SCHEMBL8918668

SCHEMBL8918668

COc1ccc2c(ccc3cnn(-c4ccc(S(C)(=O)=O)cc4)c32)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
PTGS2 P35354 13/20 0.42
PTGS1 P23219 5/20 0.41
ALDH1A1 P00352 2/20 0.41
RAB9A P51151 2/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
LRRK2 Q5S007 1/20 0.38
EGFR P00533 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9231677 0.90 CA1 (0.58) CA12CA1CA2CA9PTGS2
SCHEMBL8917550 0.78 PTGS2 (0.40) PTGS2PTGS1EGFR
SCHEMBL9229223 0.76 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8917527 0.76 PTGS2 (0.45) PTGS2PTGS1ALDH1A1
SCHEMBL8918689 0.76 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8916244 0.76 PTGS2 (0.42) PTGS2PTGS1LRRK2
SCHEMBL8920714 0.73 PTGS2 (0.46) CA12CA1CA2CA9PTGS2
SCHEMBL8918137 0.72 SLC40A1 (0.40) ALDH1A1HTR2AHTR2CKDM4E
SCHEMBL9229107 0.68 CA2 (0.53) CA12CA1CA2CA9PTGS2
SCHEMBL8920604 0.68 PTGS2 (0.46) CA12CA1CA2CA9PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed